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Cat. No. Product Name Target Signaling Pathways
T40101 (±)-1,2-Diolein

1,2-Dioleoyl-rac-glycerol,甘油1,2-二油酸酯

PKC Chromatin/Epigenetic; Cytoskeletal Signaling
(±)-1,2-Diolein (1,2-Dioleoyl-rac-glycerol) 是一种PKC 激活剂,可以增加肌小管 Ca2+内流。
T1425 Pemirolast potassium

BMY 26517,TWT-8152,吡嘧司特钾

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Pemirolast potassium (TWT-8152) 是 H1组胺受体拮抗剂和肥大细胞稳定剂,是一种具有抗过敏特性的嘧啶酮衍生物。
T15257 Etripamil

MSP-2017,(-)-MSP-2017

Calcium Channel Membrane transporter/Ion channel; Metabolism
Etripamil (MSP-2017) 是一种短效L 型钙通道拮抗剂,可用于治疗阵发性室上性心动过速的研究。它通过抑制房室结细胞中钙慢通道的钙离子流入,显示房室结传导并延长房室结不应期
T3979 Emedastine

LY188695,依美斯汀,Emadine

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Emedastine (LY188695) 是一种可口服的,选择性和高亲和力的组胺 H1受体拮抗剂,Ki 值为 1.3 nM。它是苯并咪唑衍生物,可用于过敏性鼻炎、过敏性皮肤疾病和过敏性结膜炎的研究。
T68742 Inamrinone lactate

Inamrinone lactate is a positive inotropic cardiotonic with vasodilator properties, phosphodiesterase inhibitory activity, and the ability to stimulate calcium ion influx into the cardiac cell.
T71303 Flufenamic Acid-d4

Flufenamic acid-d4 is intended for use as an internal standard for the quantification of flufenamic acid by GC- or LC-MS. Flufenamic acid is a non-steroidal anti-inflammatory drug (NSAID) and COX inhibitor (IC50s = 3 and 9.3 µM for human COX-1 and COX-2, respectively). Flufenamic acid inhibits TNF-α-induced increases in COX-2 levels and NF-κB activation in HT-29 colon cancer cells in a concentration-dependent manner. It inhibits calcium influx induced by fMLP or A23187 in human polymorphonuclear...

化合物

(±)-1,2-Diolein
Cat.No: T40101
Synonym: 1,2-Dioleoyl-rac-glycerol,甘油1,2-二油酸酯
Target: PKC
Pemirolast potassium
Cat.No: T1425
Synonym: BMY 26517,TWT-8152,吡嘧司特钾
Target: Histamine Receptor
Etripamil
Cat.No: T15257
Synonym: MSP-2017,(-)-MSP-2017
Target: Calcium Channel
Emedastine
Cat.No: T3979
Synonym: LY188695,依美斯汀,Emadine
Target: Histamine Receptor
Inamrinone lactate
Cat.No: T68742
Synonym:
Target:
Flufenamic Acid-d4
Cat.No: T71303
Synonym:
Target:
TargetMol Loading
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